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Solomon Kattar
Solomon Kattar
Verified email at merck.com
Title
Cited by
Cited by
Year
Neurofilaments consist of distinct populations that can be distinguished by C-terminal phosphorylation, bundling, and axonal transport rate in growing axonal neurites
JT Yabe, T Chylinski, FS Wang, A Pimenta, SD Kattar, MD Linsley, ...
Journal of Neuroscience 21 (7), 2195-2205, 2001
1292001
Therapeutic compounds
J Katz, J Jewell, J Jung, S Kattar, Y Hou, R MacCoss, S Ito
US Patent 8,455,477, 2013
462013
Spirocyclic compounds
SC Berk, J Close, C Hamblett, RW Heidebrecht, SD Kattar, LT Kliman, ...
US Patent 7,544,695, 2009
462009
Aminopyrimidines as Syk inhibitors
MD Altman, KL Arrington, J Burch, B Cote, JF Fournier, JY Gauthier, ...
US Patent 8,735,417, 2014
422014
Parallel medicinal chemistry approaches to selective HDAC1/HDAC2 inhibitor (SHI-1: 2) optimization
SD Kattar, LM Surdi, A Zabierek, JL Methot, RE Middleton, B Hughes, ...
Bioorganic & Medicinal Chemistry Letters 19 (4), 1168-1172, 2009
402009
Aminopyrimidines as SYK inhibitors
MD Altman, BM Andresen, KL Arrington, J Burch, KK Childers, B Cote, ...
US Patent 8,551,984, 2013
332013
Discovery of a chemical probe for PRDM9
A Allali-Hassani, MM Szewczyk, D Ivanochko, SL Organ, J Bok, JSY Ho, ...
Nature communications 10 (1), 5759, 2019
302019
Structure-guided discovery of aminoquinazolines as brain-penetrant and selective LRRK2 inhibitors
MH Keylor, A Gulati, SD Kattar, RE Johnson, RW Chau, KA Margrey, ...
Journal of medicinal chemistry 65 (1), 838-856, 2021
232021
Inhibitors of IRAK4 activity
MD Altman, JD Brubaker, ML Childers, A Donofrio, T Fischmann, ...
US Patent 9,926,330, 2018
232018
4-carboxybenzylamino derivatives as histone deacetylase inhibitors
P Harrington, S Kattar, TA Miller, MG Stanton, P Tempest, DJ Witter
US Patent 8,389,553, 2013
182013
Phosphorus derivatives as histone deacetylase inhibitors
J Close, J Grimm, RW Heidebrecht, S Kattar, TA Miller, KM Otte, ...
US Patent 7,981,874, 2011
182011
Bipyridylaminopyridines as Syk inhibitors
D Deschenes, MD Altman, JM Ellis, C Fischer, AM Haidle, SD Kattar, ...
US Patent 9,145,391, 2015
162015
Substituted pyridine spleen tyrosine kinase (SYK) inhibitors
AM Haidle, SL Knowles, SD Kattar, D Deschenes, J Burch, J Robichaud, ...
US Patent 9,376,418, 2016
152016
Aminopyrimidines as Syk inhibitors
MD Altman, KK Childers, ME Di Francesco, JM Ellis, C Fischer, J Grimm, ...
US Patent 9,290,490, 2016
152016
Spirocyclic compounds
SC Berk, J Close, C Hamblett, RW Heidebrecht, SD Kattar, LT Kliman, ...
US Patent 7,834,026, 2010
152010
Pyrazolyl derivatives as Syk inhibitors
MR Machacek, MD Altman, ET Romeo, D Vitharana, B Cash, T Siu, ...
US Patent 9,242,984, 2016
142016
Substituted diazine and triazine spleen tyrosine kinease (Syk) inhibitors
AM Haidle, MD Altman, SD Kattar, M Christopher, JM Ellis, C Fischer, ...
US Patent 9,416,111, 2016
132016
Histone deacetylase inhibitors with aryl-pyrazolyl-motifs
J Close, RW Heidebrecht, S Kattar, TA Miller, D Sloman, MG Stanton, ...
US Patent 8,026,260, 2011
132011
Optimization of brain-penetrant picolinamide derived leucine-rich repeat kinase 2 (LRRK2) inhibitors
A Gulati, CS Yeung, B Lapointe, SD Kattar, H Gunaydin, JD Scott, ...
RSC Medicinal Chemistry 12 (7), 1164-1173, 2021
112021
Substituted phenyl-Spleen Tyrosine Kinase (Syk) inhibitors
AM Haidle, J Burch, D Guay, JY Gauthier, J Robichaud, JF Fournier, ...
US Patent 9,353,066, 2016
112016
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