| Enantioselective synthesis of SM-130686 based on the development of asymmetric Cu (I) F catalysis to access 2-oxindoles containing a tetrasubstituted carbon D Tomita, K Yamatsugu, M Kanai, M Shibasaki Journal of the American Chemical Society 131 (20), 6946-6948, 2009 | 285 | 2009 |
| Total synthesis of (±)-garsubellin A A Kuramochi, H Usuda, K Yamatsugu, M Kanai, M Shibasaki Journal of the American Chemical Society 127 (41), 14200-14201, 2005 | 177 | 2005 |
| Limited brain distribution of [3R, 4R, 5S]-4-acetamido-5-amino-3-(1-ethylpropoxy)-1-cyclohexene-1-carboxylate phosphate (Ro 64-0802), a pharmacologically active form of … A Ose, M Ito, H Kusuhara, K Yamatsugu, M Kanai, M Shibasaki, ... Drug Metabolism and Disposition 37 (2), 315-321, 2009 | 143 | 2009 |
| 26Q-am155 K Yamatsugu, L Yin, S Kamijo, Y Kimura, M Kanai, M Shibasaki Angew. Chem. Int. Ed, 48, 2009 | 140 | 2009 |
| A concise synthesis of Tamiflu: third generation route via the Diels–Alder reaction and the Curtius rearrangement K Yamatsugu, S Kamijo, Y Suto, M Kanai, M Shibasaki Tetrahedron letters 48 (8), 1403-1406, 2007 | 117 | 2007 |
| P-glycoprotein restricts the penetration of oseltamivir across the blood-brain barrier A Ose, H Kusuhara, K Yamatsugu, M Kanai, M Shibasaki, T Fujita, ... Drug Metabolism and Disposition 36 (2), 427-434, 2008 | 104 | 2008 |
| Synthetic posttranslational modifications: chemical catalyst-driven regioselective histone acylation of native chromatin Y Amamoto, Y Aoi, N Nagashima, H Suto, D Yoshidome, Y Arimura, ... Journal of the American Chemical Society 139 (22), 7568-7576, 2017 | 71 | 2017 |
| Intermolecular stereoselective iridium-catalyzed allylic alkylation: an evolutionary account SE Shockley, JC Hethcox, BM Stoltz Synlett 29 (19), 2481-2492, 2018 | 54 | 2018 |
| Oseltamivir enhances hippocampal network synchronization A Usami, T Sasaki, N Satoh, T Akiba, S Yokoshima, T Fukuyama, ... Journal of pharmacological sciences 106 (4), 659-662, 2008 | 45 | 2008 |
| Recent development in synthetic strategies for oseltamivir phosphate M Shibasaki, M Kanai, K Yamatsugu Israel Journal of Chemistry 51 (3‐4), 316-328, 2011 | 41 | 2011 |
| An alternative synthesis of Tamiflu®: a synthetic challenge and the identification of a ruthenium-catalyzed dihydroxylation route K Yamatsugu, M Kanai, M Shibasaki Tetrahedron 65 (31), 6017-6024, 2009 | 41 | 2009 |
| Nuclear envelope expansion is crucial for proper chromosomal segregation during a closed mitosis A Takemoto, SA Kawashima, JJ Li, L Jeffery, K Yamatsugu, O Elemento, ... Journal of cell science 129 (6), 1250-1259, 2016 | 40 | 2016 |
| LC–MS/MS-based quantitative study of the acyl group-and site-selectivity of human sirtuins to acylated nucleosomes K Tanabe, J Liu, D Kato, H Kurumizaka, K Yamatsugu, M Kanai, ... Scientific reports 8 (1), 2656, 2018 | 38 | 2018 |
| Synthetic chromatin acylation by an artificial catalyst system T Ishiguro, Y Amamoto, K Tanabe, J Liu, H Kajino, A Fujimura, Y Aoi, ... Chem 2 (6), 840-859, 2017 | 34 | 2017 |
| Two approaches toward the formal total synthesis of oseltamivir phosphate (Tamiflu): Catalytic enantioselective three-component reaction strategy and l-glutamic acid strategy K Alagiri, M Furutachi, K Yamatsugu, N Kumagai, T Watanabe, ... The Journal of Organic Chemistry 78 (8), 4019-4026, 2013 | 32 | 2013 |
| Live-cell epigenome manipulation by synthetic histone acetylation catalyst system Y Fujiwara, Y Yamanashi, A Fujimura, Y Sato, T Kujirai, H Kurumizaka, ... Proceedings of the National Academy of Sciences 118 (4), e2019554118, 2021 | 28 | 2021 |
| Catalytic Chemoselective O-Phosphorylation of Alcohols K Domon, M Puripat, K Fujiyoshi, M Hatanaka, SA Kawashima, ... ACS Central Science 6 (2), 283-292, 2020 | 28 | 2020 |
| A method for the synthesis of an oseltamivir PET tracer M Morita, T Sone, K Yamatsugu, Y Sohtome, S Matsunaga, M Kanai, ... Bioorganic & medicinal chemistry letters 18 (2), 600-602, 2008 | 23 | 2008 |
| Leading approaches in synthetic epigenetics for novel therapeutic strategies K Yamatsugu, SA Kawashima, M Kanai Current Opinion in Chemical Biology 46, 10-17, 2018 | 22 | 2018 |
| Synthesis of Malononitrile-Substituted Diarylmethines via 1, 6-Addition of Masked Acyl Cyanides to para-Quinone Methides K Zhao, Y Zhi, A Wang, D Enders Synthesis 50 (04), 872-880, 2018 | 22 | 2018 |
