| Liposome/water lipophilicity: methods, information content, and pharmaceutical applications GP van Balen, CM Martinet, G Caron, G Bouchard, M Reist, PA Carrupt, ... Medicinal research reviews 24 (3), 299-324, 2004 | 187 | 2004 |
| Impact of dynamically exposed polarity on permeability and solubility of chameleonic drugs beyond the rule of 5 M Rossi Sebastiano, BC Doak, M Backlund, V Poongavanam, B Over, ... Journal of medicinal chemistry 61 (9), 4189-4202, 2018 | 177 | 2018 |
| Lipophilicity profiles of ampholytes A Pagliara, PA Carrupt, G Caron, P Gaillard, B Testa Chemical reviews 97 (8), 3385-3400, 1997 | 175 | 1997 |
| Ligand specificity of the genetic variants of human α1-acid glycoprotein: generation of a three-dimensional quantitative structure-activity relationship model for drug binding … F Hervé, G Caron, JC Duché, P Gaillard, NA Rahman, ... Molecular Pharmacology 54 (1), 129-138, 1998 | 121 | 1998 |
| Structure‐Lipophilicity Relationships of Neutral and Protonated β‐Blockers, Part I, Intra‐ and Intermolecular Effects in Isotropic Solvent Systems G Caron, G Steyaert, A Pagliara, F Reymond, P Crivori, P Gaillard, ... Helvetica Chimica Acta 82 (8), 1211-1222, 1999 | 109 | 1999 |
| Combined molecular lipophilicity descriptors and their role in understanding intramolecular effects G Caron, F Reymond, PA Carrupt, HH Girault, B Testa Pharmaceutical science & technology today 2 (8), 327-335, 1999 | 109 | 1999 |
| Molecular Factors Influencing Retention on Immobilized Artificial Membranes (IAM) Compared to Partitioning in Liposomes and n-Octanol A Taillardat-Bertschinger, CAM Martinet, PA Carrupt, M Reist, G Caron, ... Pharmaceutical research 19, 729-737, 2002 | 108 | 2002 |
| Intramolecular hydrogen bonding: An opportunity for improved design in medicinal chemistry G Caron, J Kihlberg, G Ermondi Medicinal Research Reviews 39 (5), 1707-1729, 2019 | 105 | 2019 |
| Lipophilicity behavior of model and medicinal compounds containing a suilfide, sulfoxide, or sulfone moiety G Caron, P Gaillard, PA Carrupt, B Testa Helvetica chimica acta 80 (2), 449-462, 1997 | 102 | 1997 |
| Integrating intramolecular hydrogen bonding (IMHB) considerations in drug discovery using ΔlogP as a tool M Shalaeva, G Caron, YA Abramov, TN O’Connell, MS Plummer, ... Journal of medicinal chemistry 56 (12), 4870-4879, 2013 | 94 | 2013 |
| Conformational sampling of macrocyclic drugs in different environments: can we find the relevant conformations? V Poongavanam, E Danelius, S Peintner, L Alcaraz, G Caron, ... ACS omega 3 (9), 11742-11757, 2018 | 84 | 2018 |
| Molecular and statistical modeling of reduction peak potential and lipophilicity of platinum (IV) complexes JA Platts, G Ermondi, G Caron, M Ravera, E Gabano, L Gaviglio, G Pelosi, ... JBIC Journal of Biological Inorganic Chemistry 16, 361-372, 2011 | 74 | 2011 |
| N‐substituted analogues of S‐nitroso‐N‐acetyl‐D,L‐penicillamine: chemical stability and prolonged nitric oxide mediated vasodilatation in isolated rat femoral … IL Megson, S Morton, IR Greig, FA Mazzei, RA Field, AR Butler, G Caron, ... British journal of pharmacology 126 (3), 639-648, 1999 | 65 | 1999 |
| On the complexation of quercetin with methyl-β-cyclodextrin: photostability and antioxidant studies ME Carlotti, S Sapino, E Ugazio, G Caron Journal of Inclusion Phenomena and Macrocyclic Chemistry 70, 81-90, 2011 | 64 | 2011 |
| Mechanisms of liposomes/water partitioning of (p-methylbenzyl) alkylamines R Fruttero, G Caron, E Fornatto, D Boschi, G Ermondi, A Gasco, ... Pharmaceutical research 15, 1407-1413, 1998 | 64 | 1998 |
| Contribution of ionization and lipophilicity to drug binding to albumin: a preliminary step toward biodistribution prediction G Ermondi, M Lorenti, G Caron Journal of medicinal chemistry 47 (16), 3949-3961, 2004 | 62 | 2004 |
| Glycosylated copper (II) ionophores as prodrugs for β-glucosidase activation in targeted cancer therapy V Oliveri, M Viale, G Caron, C Aiello, R Gangemi, G Vecchio Dalton Transactions 42 (6), 2023-2034, 2013 | 61 | 2013 |
| Glycosylated copper (II) ionophores as prodrugs for β-glucosidase activation in targeted cancer therapy V Oliveri, M Viale, G Caron, C Aiello, R Gangemi, G Vecchio Dalton Transactions 42 (6), 2023-2034, 2013 | 61 | 2013 |
| Flexibility in early drug discovery: focus on the beyond-Rule-of-5 chemical space G Caron, V Digiesi, S Solaro, G Ermondi Drug Discovery Today 25 (4), 621-627, 2020 | 58 | 2020 |
| Molecular descriptors for polarity: the need for going beyond polar surface area G Caron, G Ermondi Future Medicinal Chemistry 8 (17), 2013-2016, 2016 | 57 | 2016 |
Giuseppe ErmondiUniversity of TorinoGeverifieerd e-mailadres voor unito.it
